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ER degrader 2

CAT: 0804-HY-142926Size: 1 EachDry Ice: NoHazardous: No
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CAT#:0804-HY-142926Size:1 Each
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
ER degrader 2 is a potent degrader of estrogen receptor (ER) . The estrogen signaling system plays an important role in regulating cell growth, differentiation and apoptosis. ER degrader 2 has the potential for the research of cancer diseases (extracted from patent CN112830919A, compound 1) [1].
CAS Number
2390147-41-6
UNSPSC
12352005
Target
Estrogen Receptor/ERR
Type
Reference compound
Related Pathways
Vitamin D Related/Nuclear Receptor
Applications
Cancer-programmed cell death
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/er-degrader-2.html
Solubility
10 mM in DMSO
Smiles
CC(C)(F)CN1[C@@](C2=C(C=C(C=C2F)OCCNC/C=C/C(N3CCOCC3)=O)F)([H])C4=CC=C(C5=CN(N=C5)C)C=C4C[C@H]1C
Molecular Formula
C34H42F3N5O3
Molecular Weight
625.72
References & Citations
[1]Miaomiao Zhao, et al. Benzopiperidine derivatives pharmaceutically available salts and methods for their preparation. Patent CN112830919A.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported