ER degrader 1

ER degrader 1

• CAS Number: 2667015-33-8
• UNSPSC Description: ER degrader 1 is a potent degrader of estrogen receptor (ER). The estrogen signaling system plays an important role in regulating cell growth, differentiation and apoptosis. ER degrader 1 has the potential for the research of cancer diseases (extracted from patent WO2021139756A1, compound 11)[1].
• Target Antigen: Estrogen Receptor/ERR
• Type: Reference compound
• Related Pathways: Vitamin D Related/Nuclear Receptor
• Applications: Cancer-programmed cell death
• Field of Research: Cancer
• Assay Protocol: https://www.medchemexpress.com/er-degrader-1.html
• Solubility: 10 mM in DMSO
• Smiles: OCC(F)(F)CN1[C@@](C2=C(C=C(C=N2)N[C@@H]3CN(CC3)CCCF)F)([H])C4=C(C[C@H]1C)C=C5C(OCO5)=C4
• Molecular Weight: 524.55
• References & Citations: [1]Fanglong Yang, et al. Tricyclic tetrahydroisoquinoline derivatives, their preparation methods and their application in medicine. Patent WO2021139756A1.
• Shipping Conditions: Room temperature
• Clinical Information: No Development Reported