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ER degrader 3

CAT: 0804-HY-142927Size: 1 EachDry Ice: NoHazardous: No
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CAT#:0804-HY-142927Size:1 Each
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Description
ER degrader 3 is a potent degrader of estrogen receptor (ER) . The estrogen signaling system plays an important role in regulating cell growth, differentiation and apoptosis. ER degrader 3 has the potential for the research of cancer diseases (extracted from patent WO2018233591A1, compound 1) [1].
CAS Number
2254818-47-6
UNSPSC
12352005
Target
Estrogen Receptor/ERR
Type
Reference compound
Related Pathways
Vitamin D Related/Nuclear Receptor
Applications
Cancer-programmed cell death
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/er-degrader-3.html
Solubility
10 mM in DMSO
Smiles
NCCCC[C@H](N)C(O)=O.C[C@H]1N(C2=CC=C(C3CC3)C=C2)[C@@](C4=CC=C(C=C4)/C=C/C(O)=O)([H])C5=CC=C(C6=CN(N=C6)CC)C=C5C1
Molecular Formula
C39H47N5O4
Molecular Weight
649.82
References & Citations
[1]Lingfeng You, et al. A kind of salt of benzopiperidine derivatives, its crystal form and salt, the preparation method of its crystal form. Patent WO2018233591A1.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported

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