AR Degrader-1
- Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
- Dry Ice Shipment: No


AR Degrader-1
Target :
Molecular Glues|||Androgen Receptor|||E1/E2/E3 EnzymeRelated Pathways :
Endocrinology/Hormones|||Ubiquitination|||PROTACBioactivity :
AR Degrader-1 (Compound ML 2-9) is a monovalent degrader of androgen receptors (AR) categorized under molecular glues. In LNCaP prostate cancer cells, it facilitates AR degradation through DCAF16 (E3 ligase) while exhibiting minimal cytotoxicity.Molecular Formula :
C24H27ClN6O4SShipping Conditions :
Cool packStorage Temperature :
-20°C

