Products for Research Use Only

PDE4-IN-17

CAT: 0931-T210238-01Size: 10 mgDry Ice: NoHazardous: No
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CAT#:0931-T210238-01Size:10 mg
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Target
PDE
Related Pathways
Metabolism
Bioactivity
PDE4-IN-17 (compound 4e) is a potent PDE4 inhibitor. It effectively inhibits PDE4B and PDE4D with IC50 values of 10.0 nM and 15.2 nM, respectively. In SD rats, PDE4-IN-17 demonstrates good oral bioavailability (F=66%) and a relatively long half-life (t1/2=2.0 h) .
Molecular Formula
C17H16N2O3
Shipping Conditions
Ice Packs
Storage Temperature
-20°C