Products for Research Use Only

AR Degrader-1

CAT: 0013-GTR19262513-01Size: 50 mgDry Ice: NoHazardous: No
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CAT#:0013-GTR19262513-01Size:50 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
AR Degrader-1 (Compound ML 2-9) is a monovalent degrader of androgen receptors (AR) categorized under molecular glues. In LNCaP prostate cancer cells, it facilitates AR degradation through DCAF16 (E3 ligase) while exhibiting minimal cytotoxicity.
Field of Research
Metabolism Research, Pharmacology & Drug Discovery, Protein Biochemistry
Molecular Formula
C24H27ClN6O4S
Storage Conditions
-20°C
Notes
For research use only.