Products for Research Use Only

PROTAC AR-NTD degrader 1

CAT: 0013-GTR19230908-01Size: 5 mgDry Ice: NoHazardous: No
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CAT#:0013-GTR19230908-01Size:5 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
PROTAC AR-NTD antagonist 1 is a heterobifunctional degrader that selectively targets the AR-V7 splice variant via its N-terminal domain. It induces potent AR-V7 degradation and apoptosis in prostate cancer cell lines, such as VCaP, and serves as a key tool for investigating castration-resistant prostate cancer mechanisms in vitro.
Field of Research
Cell Biology, Metabolism Research, Stem Cell & Developmental Biology
Molecular Formula
C41H47ClN6O7
Molecular Weight
771.3
Storage Conditions
-20°C
Notes
For research use only.