PRMT5-MTA-IN-2

• UNSPSC Description:

  PRMT5-MTA-IN-2 (compund 1) is a MTA co-inhibitor of PRMT5 with IC50 less than 1.5 nM[1].

• Target Antigen:

  Histone Methyltransferase

• Type:

  Reference compound

• Related Pathways:

  Epigenetics

• Applications:

  Cancer-programmed cell death

• Field of Research:

  Cancer

• Assay Protocol:

  https://www.medchemexpress.com/prmt5-mta-in-2.html

• Smiles:

  NC1=NC2=C(C3=C1COC3)NC(C(N([C@@H]4CCCC5=CC=CN=C54)CC6=NC=C(C=C6)C7=C(C=NC=C7F)F)=O)=C2

• Molecular Weight:

  553.56

• References & Citations:

  [1]WO2024199255A1

• Shipping Conditions:

  Room temperature

• Clinical Information:

  No Development Reported