PDE4-IN-10

CAT:
931-T60346-01
Size:
25 mg
  • Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
  • Dry Ice Shipment: No
PDE4-IN-10 - image 1

PDE4-IN-10

  • Target:

    Others|||PDE|||TNF
  • Related Pathways:

    Metabolism|||Apoptosis|||Others
  • Bioactivity:

    PDE4-IN-10 (compound 7a) is a potent PDE4 inhibitor with an IC50 of 7.01 ?M for PDE4B, demonstrating selectivity, microsomal stability, TNF-? inhibition, and no major toxicities in vitro [1].
  • Smiles:

    CC1=CC2=C(C=3C1=CC=CC3)N=CC=4C2=CC=CC4
  • Molecular Formula:

    C18H13N
  • Molecular Weight:

    243.3
  • Shipping Conditions:

    Cool pack
  • Storage Temperature:

    -20°C
  • CAS Number:

    2413564-66-4