LPAR1 antagonist 2

• UNSPSC Description:

  LPAR1 antagonist 2 (example 76) is an LPAR1 antagonist with an average IC50 of 130 nM[1].

• Target Antigen:

  LPL Receptor

• Type:

  Reference compound

• Related Pathways:

  GPCR/G Protein

• Field of Research:

  Others

• Assay Protocol:

  https://www.medchemexpress.com/lpar1-antagonist-2.html

• Solubility:

  10 mM in DMSO

• Smiles:

  O=C(C1=CC=C(CN(CC)C(C2=CC=C(C=C2)OC3=C(Cl)C=CC=C3)=O)C=C1)O

• Molecular Weight:

  409.86

• References & Citations:

  [1]Preparation of amide derivatives as lysophosphatidic acid receptor antagonists. World Intellectual Property Organization, et al. World Intellectual Property Organization, WO2015025164 A1 2015-02-26.

• Shipping Conditions:

  Room temperature

• Clinical Information:

  No Development Reported

• CAS Number:

  1664336-46-2