P-gp modulator 2
- Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
- Dry Ice Shipment: No


P-gp modulator 2
UNSPSC Description:
P-gp modulator 2 (Compound 27) is a potent, competitive, allosteric P-glycoprotein (P-gp) modulator[1].Target Antigen:
P-glycoproteinType:
Reference compoundRelated Pathways:
Membrane Transporter/Ion ChannelApplications:
Cancer-programmed cell deathField of Research:
CancerAssay Protocol:
https://www.medchemexpress.com/p-gp-modulator-2.htmlSolubility:
10 mM in DMSOSmiles:
COC1=CC=C(C=C1)[C@@H]2C/C(C3=C(O2)C=C(C=C3O)OC)=N\NC4=CC=C(C=N4)BrMolecular Weight:
470.32References & Citations:
[1]Ferreira RJ, et al. Nitrogen-containing naringenin derivatives for reversing multidrug resistance in cancer. Bioorg Med Chem. 2020 Dec 1;28(23):115798.Shipping Conditions:
Room temperatureClinical Information:
No Development ReportedCAS Number:
2987145-05-9
