KAT modulator-1
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- Dry Ice Shipment: No


KAT modulator-1
UNSPSC Description:
KAT modulator-1 (Compound 3) is a KAT modulator. KAT modulator-1 can interact with p300 full-length but not with the catalytic domain. KAT modulator-1 can be used for epigenetics research[1].Target Antigen:
Histone AcetyltransferaseType:
Reference compoundRelated Pathways:
EpigeneticsApplications:
Cancer-programmed cell deathField of Research:
CancerAssay Protocol:
https://www.medchemexpress.com/kat-modulator-1.htmlSolubility:
DMSO : 100 mg/mL (ultrasonic;warming;heat to 80°C)Smiles:
O=C(C)/C(C(C)=O)=C/CCCCCCCCCCCCCCMolecular Weight:
308.50References & Citations:
[1]Milite C, et al. Modulation of the activity of histone acetyltransferases by long chain alkylidenemalonates (LoCAMs). Bioorg Med Chem. 2011 Jun 15;19(12):3690-701.Shipping Conditions:
Room TemperatureClinical Information:
No Development ReportedCAS Number:
1314006-43-3
