GPR17 modulator-1

• Description :

  GPR17 modulator-1 (Compound 2-046) is a modulator for G protein-coupled receptor 17 GPR17, with an IC50hGPR17 in CHO. GPR17 modulator-1 exhibits moderate pharmacokinetic characteristics in mice. GPR17 modulator-1 ix blood-brain barrier (BBB) permeable[1].

• CAS Number :

  [3039853-91-0]

• UNSPSC :

  12352005

• Target :

  Transmembrane Glycoprotein

• Type :

  Reference compound

• Related Pathways :

  Immunology/Inflammation

• Applications :

  Neuroscience-Neuromodulation

• Field of Research :

  Neurological Disease

• Assay Protocol :

  https://www.medchemexpress.com/gpr17-modulator-1.html

• Smiles :

  O=S(NC1=CC(F)=C(OCC(F)F)N=C1OC)(C2=C3C=CC(Cl)=CN3N=C2)=O

• Molecular Formula :

  C15H12ClF3N4O4S

• Molecular Weight :

  436.79

• References & Citations :

  [1]Han X, et al., Gpr17 modulators and uses thereof. WO2024104462.

• Shipping Conditions :

  Room temperature

• Scientific Category :

  Reference compound1

• Clinical Information :

  No Development Reported