GPR17 modulator-1

• Bioactivity :

  GPR17 Modulator-1 (Compound 2-046) is a regulator of the G protein-coupled receptor 17 (GPR17), displaying an IC50 of less than 10 nM against hGPR17 in CHO cells. This compound exhibits moderate pharmacokinetic properties in mice and possesses the ability to permeate the blood-brain barrier (BBB) .

• Smiles :

  O=S(=O)(NC1=CC(F)=C(N=C1OC)OCC(F)F)C=2C=NN3C=C(Cl)C=CC23

• Molecular Formula :

  C15H12ClF3N4O4S

• Molecular Weight :

  436.79

• Shipping Conditions :

  Cool pack

• Storage Temperature :

  -20°C

• CAS Number :

  3039853-91-0