Integrin modulator 1
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Integrin modulator 1
UNSPSC Description:
Integrin modulator 1 is a potent and selective α4β1 integrin agonist, with an IC50 of 9.8 nM for RGD-binding α4β1. Integrin modulator 1 increases cell adhesion mediated by α4β1 integrin, with an EC50 of 12.9 nM[1].Target Antigen:
IntegrinType:
Reference compoundRelated Pathways:
CytoskeletonField of Research:
Inflammation/ImmunologyAssay Protocol:
https://www.medchemexpress.com/integrin-modulator-1.htmlSmiles:
O=C(CC(N1C(NC2=CC=CC=C2C)=O)CC1=O)OMolecular Weight:
262.26References & Citations:
[1]Baiula M, et, al. New β-Lactam Derivatives Modulate Cell Adhesion and Signaling Mediated by RGD-Binding and Leukocyte Integrins. J Med Chem. 2016 Nov 10;59(21):9721-9742.Shipping Conditions:
Room TemperatureCAS Number:
2023788-32-9
