Kinase modulator-1

CAT: 0931-MF-0119351-01Size: 10 mgDry Ice: NoHazardous: No
CAT#:0931-MF-0119351-01Size:10 mg
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AVAILABILITY: InStock
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
927697-17-4
Target
Bcr-Abl
Related Pathways
Angiogenesis|||Tyrosine Kinase/Adaptors|||Cytoskeletal Signaling
Bioactivity
Kinase modulator-1 (P142, MS: m/z 445) is a kinase regulator that inhibits Bcr-Abl activity, specifically targeting drug-resistant mutant kinases such as T315IBcr-Abl. It is applicable for research in cancers like chronic myeloid leukemia (CML) .
Smiles
O=C(OC)NC=1C=CC(=CC1C(=O)N(C)C)C2=CN=C3NC=C(C=4C=CC=CC4OC)C3=C2
Molecular Formula
C25H24N4O4
Molecular Weight
444.48
Shipping Conditions
Cool pack
Storage Temperature
-20°C

Alternative Products

CatalogName
HY-177273Kinase modulator-1
MBS623273-01Hematopoietic Progenitor Kinase 1 (HPK1, Mitogen-activated Protein Kinase Kinase Kinase Kinase 1, MAP4K1, MAPK/ERK Kinase Kinase Kinase 1, MEK Kinase Kinase 1, MEKKK 1)
228331PXK (PX Serine/Threonine Kinase, PX Ser/Thr Kinase v2, Modulator of Na, K-ATPase, MONaKA) discontinued
MBS6004364-01MAP4K1 (Mitogen-activated Protein Kinase Kinase Kinase Kinase 1, MAPK/ERK Kinase Kinase Kinase 1, MEK Kinase Kinase 1, MEKKK 1, Hematopoietic Progenitor Kinase, HPK1)
319519-01HPK1 (MAP4K1, Mitogen-activated protein kinase kinase kinase kinase 1, Hematopoietic progenitor kinase, MAPK/ERK kinase kinase kinase 1, MEK kinase kinase 1, MEKKK 1)
323584MAP4K1 (Mitogen-activated protein kinase kinase kinase kinase 1, EC 2.7.11.1, MAPK/ERK kinase kinase kinase 1, MEK kinase kinase 1, MEKKK 1)
150067MAP4K1 (Mitogen-activated Protein Kinase Kinase Kinase Kinase 1, MAPK/ERK Kinase Kinase Kinase 1, MEK Kinase Kinase 1, MEKKK 1, Hematopoietic Progenitor Kinase, HPK1) discontinued
MBS628049-01MAP4K1, CT (Mitogen-activated Protein Kinase Kinase Kinase Kinase 1, MAPK/ERK Kinase Kinase Kinase 1, MEK Kinase Kinase 1, MEKKK 1, Hematopoietic Progenitor Kinase, HPK1)
H1827-59B-PHematopoietic Progenitor Kinase 1, Control Peptide (HPK1, Mitogen-activated Protein Kinase Kinase Kinase Kinase 1, MAP4K1, MAPK/ERK Kinase Kinase Kinase 1, MEK Kinase Kinase 1, MEKKK 1) discontinued
MBS6488246-01MAP4K1, CT (Mitogen-activated Protein Kinase Kinase Kinase Kinase 1, MAPK/ERK Kinase Kinase Kinase 1, MEK Kinase Kinase 1, MEKKK 1, Hematopoietic Progenitor Kinase, HPK1) (AP)

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