PL-017

CAT: 0931-TP1958Size: 10 mgDry Ice: NoHazardous: No
CAT#:0931-TP1958Size:10 mg
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AVAILABILITY: InStock
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
83397-56-2
Target
Opioid Receptor
Related Pathways
GPCR/G Protein|||Neuroscience|||Endocrinology/Hormones
Bioactivity
Selective ? opioid receptor agonist (IC50 values are 5.5 and > 10000 nM for inhibition of 125I-FK 33,824 and 125I-DADLE binding to ? and ? sites respectively) . Produces naloxone-reversible analgesia, catalepsy and hyperthermia following central administration in rats in vivo.
Smiles
C(N([C@H](C(=O)N1[C@@H](C(N)=O)CCC1)CC2=CC=CC=C2)C)(=O)[C@H]3N(C([C@H](CC4=CC=C(O)C=C4)N)=O)CCC3
Molecular Formula
C29H37N5O5
Molecular Weight
535.64
Shipping Conditions
Cool pack
Storage Temperature
-20°C