PL-017

CAT: 0804-HY-P1338Size: 1 EachDry Ice: NoHazardous: No
CAT#:0804-HY-P1338Size:1 Each
Selected
PRICE
AVAILABILITY: InStock
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
Product image 1
1 / 1
Description
PL-017 is a potent and selective μ opioid receptor agonist with an IC50 of 5.5 nM for 125I-FK 33,824 binding to μ site. PL-017 produces long-lasting, reversible analgesia in rats[1].
CAS Number
[83397-56-2]
UNSPSC
12352209
Target
Opioid Receptor
Type
Peptides
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/pl-017.html
Solubility
H2O
Smiles
O=C(N1[C@H](CCC1)C(N)=O)[C@H](CC2=CC=CC=C2)N(C)C([C@H]3N(CCC3)C([C@@H](N)CC4=CC=C(O)C=C4)=O)=O
Molecular Formula
C29H37N5O5
Molecular Weight
535.63
References & Citations
[1]K J Chang, et al. Potent morphiceptin analogs: structure activity relationships and morphine-like activities. J Pharmacol Exp Ther. 1983 Nov;227 (2) :403-8.
Shipping Conditions
Room temperature
Scientific Category
Peptides
Clinical Information
No Development Reported
Isoform
μ Opioid Receptor/MOR

Related Products

CatalogName
HY-W419140-01AND-017
HY-121642SL-017
HY-174212MXC-017
HY-18051CXL 017
HY-147082-01GA-017
HY-118821JTC-017
HY-19291DL-017
HY-171715PL-13
HY-137798-01Chromozym PL
HY-P3562PL-3994

Alternative Products

CatalogName
M30590-01PL 017
MF-0109880PL-017
MBS5817824PL-017 TFA
MF-0052216-01JTC-017
BA9120-10GA-017
MF-0118080-01MXC-017
MF-0039443SL-017
E7970-01ε-PL
S8708-25mgAZD0364 (ATG-017)

Popular Products