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BMS-196085

CAT: 0804-HY-120223Size: 1 EachDry Ice: NoHazardous: No
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CAT#:0804-HY-120223Size:1 Each
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Description
BMS-196085 is an orally active, potent and selective full agonist against human β3 adrenergic receptor with a Ki value of 21 nM. BMS-196085 also has partial agonist activity at the β1 receptor. BMS-196085 is promising for research of obesity and type-II diabetes[1][2].
CAS Number
170686-10-9
UNSPSC
12352005
Target
Adrenergic Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Metabolism-protein/nucleotide metabolism
Field of Research
Metabolic Disease
Assay Protocol
https://www.medchemexpress.com/bms-196085.html
Smiles
O[C@H](C1=CC(NS(C)(=O)=O)=C(C=C1)O)CN[C@@H](C2=CC=C(C=C2)OC(F)F)CC3=CC=CC=C3
Molecular Formula
C24H26F2N2O5S
Molecular Weight
492.54
References & Citations
[1]Gavai A V, et al. BMS-196085: a potent and selective full agonist of the human β3 adrenergic receptor[J]. Bioorganic & medicinal chemistry letters, 2001, 11 (23) : 3041-3044.|[2]Hu B, et al. Orally bioavailable β3-adrenergic receptor agonists as potential therapeutic agents for obesityand type-II diabetes[J]. Progress in medicinal chemistry, 2003, 41: 167-194.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
Phase 1

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