RLH-033

• Description :

  RLH-033 is a potent and selective ligand for the sigma 1 recognition site. RLH-033 has high affinity for sigma 1 sites labeled by [3H] (+) -pentazocine with a Ki of 50 pM[1].

• UNSPSC :

  12352005

• Target :

  MAChR

• Type :

  Reference compound

• Related Pathways :

  GPCR/G Protein; Neuronal Signaling

• Applications :

  Neuroscience-Neuromodulation

• Field of Research :

  Neurological Disease

• Assay Protocol :

  https://www.medchemexpress.com/rlh-033.html

• Solubility :

  10 mM in DMSO

• Smiles :

  O=C(OCCN1CCC(CC1)C2=CC=CC=C2)C3(CCCC3)C4=CC=C(C=C4)[N+]([O-])=O.[H]Cl

• Molecular Formula :

  C25H31ClN2O4

• Molecular Weight :

  458.98

• References & Citations :

  [1]R L Hudkins, et al. RLH-033, a novel, potent and selective ligand for the sigma 1 recognition site. Eur J Pharmacol. 1994 Dec 12;271 (1) :235-6.

• Shipping Conditions :

  Room temperature

• Scientific Category :

  Reference compound1

• Clinical Information :

  No Development Reported

• CAS Number :

  [157097-10-4]