ER-819762

CAT: 0804-HY-116099-01Size: 1 mgDry Ice: NoHazardous: No
CAT#:0804-HY-116099-01Size:1 mg
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Description
ER-819762 is an orally active, highly selective prostaglandin E2 (PGE2) EP4 receptor antagonist with an EC50 of 70 nM against human EP4 receptor. ER-819762 can be used for rheumatoid arthritis research[1].
CAS Number
[1155773-15-1]
UNSPSC
12352005
Target
Prostaglandin Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein
Applications
COVID-19-immunoregulation
Field of Research
Inflammation/Immunology
Assay Protocol
https://www.medchemexpress.com/er-819762.html
Solubility
10 mM in DMSO
Smiles
CCN1C2(CCN(CC2)CC3=CC(C)=CC(C)=C3)C(N(CC4=CC(OC)=C5)C1=O)=C[C@H](C)C4=C5OC
Molecular Formula
C30H39N3O3
Molecular Weight
489.65
References & Citations
[1]Chen Q, et al. A novel antagonist of the prostaglandin E (2) EP (4) receptor inhibits Th1 differentiation and Th17 expansion and is orally active in arthritis models. Br J Pharmacol. 2010 May;160 (2) :292-310.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
EP

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