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Erα-IN-1

CAT: 0804-HY-168644Size: 1 EachDry Ice: NoHazardous: No
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CAT#:0804-HY-168644Size:1 Each
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
Erα-IN-1 (compound 3c) is an inhibitor of estrogen receptor α (ERα), blocking ERa activity in MCF7/ERE-LUC cells.[1].
UNSPSC
12352005
Target
Estrogen Receptor/ERR
Type
Reference compound
Related Pathways
Vitamin D Related/Nuclear Receptor
Applications
Metabolism-protein/nucleotide metabolism
Field of Research
Endocrinology
Assay Protocol
https://www.medchemexpress.com/erα-in-1.html
Smiles
CC1=NC2=C(C=CC(F)=C2)C3=C1C4=CC=CC=C4N3
Molecular Formula
C16H11FN2
Molecular Weight
250.27
References & Citations
[1]Bogdanov FB, et al. Photochemical Metal-Free synthesis and biological Assessment of isocryptolepine analogues targeting estrogen receptor Alpha in breast cancer cells. Bioorg Chem. 2024 Dec;153:107942.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported

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