BMT-124110 (formic)

CAT: 0804-HY-135871A-01Size: 1 mgDry Ice: NoHazardous: No
CAT#:0804-HY-135871A-01Size:1 mg
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Description
BMT-124110 formic is a potent, selective AAK1 inhibitor, with an IC50 of 0.9 nM. BMT-124110 shows antinociceptive activity. BMT-124110 formic inhibits BMP-2-inducible protein kinase (BIKE) and Cyclin G-associated kinase (GAK) with IC50s of 17 and 99 nM, respectively[1].
UNSPSC
12352005
Target
AAK1
Related Pathways
Neuronal Signaling
Field of Research
Neurological Disease
Purity
99.17
Smiles
CC(NC1=CC2=C(COC3=CC(OC[C@@](C)(N)CC(C)C)=CC=C32)C=N1)=O.OC=O
Molecular Formula
C22H29N3O5
Molecular Weight
415.48
References & Citations
[1]Kostich W, et al. Inhibition of AAK1 Kinase as a Novel Therapeutic Approach to Treat Neuropathic Pain. J Pharmacol Exp Ther. 2016 Sep;358 (3) :371-86.
Shipping Conditions
Room Temperature
Storage Conditions
4°C (Powder, sealed storage, away from moisture)
Scientific Category
Reference compound1
Clinical Information
No Development Reported

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