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Antitumor agent-123

CAT: 0931-T208233-01Size: 10 mgDry Ice: NoHazardous: No
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CAT#:0931-T208233-01Size:10 mg
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Target
HDAC, JAK
Related Pathways
Chromatin/Epigenetic, Angiogenesis, Stem Cells, Tyrosine Kinase/Adaptors, JAK/STAT signaling, DNA Damage/DNA Repair
Bioactivity
Antitumor agent-123 (Compound 4d) effectively inhibits various kinase targets with anticancer properties, including JAK2, JAK3, HDAC1, and HDAC6, with IC50 values of 34.6 μM for JAK2 and 2.6 μM for JAK3. In solid tumor models, Antitumor agent-123 demonstrates moderate activity.
Molecular Formula
C19H14ClFN6O2
Shipping Conditions
Ice Packs
Storage Temperature
-20°C