CK-963
- Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
- Dry Ice Shipment: No


CK-963
UNSPSC Description:
CK-963 is an activator for cardiac troponin (cTnC) with Ki of 11.5 μM. CK-963 exhibits activity in enhancing cardiac contractility in Sprague-Dawley rats[1].Target Antigen:
OthersType:
Reference compoundRelated Pathways:
OthersApplications:
Neuroscience-NeuromodulationField of Research:
Cardiovascular DiseaseAssay Protocol:
https://www.medchemexpress.com/ck-963.htmlSolubility:
DMSO : 100 mg/mL (ultrasonic)Smiles:
O=S(C(C=C(C(NC(C)=N1)=O)C1=C2)=C2OCCN3CCOCC3)(NC4=CC=C(N5C[C@H](C)C[C@@H](C)C5)N=C4)=OMolecular Weight:
556.68References & Citations:
[1]Collibee SE, et al., Cardiac Troponin Activator CK-963 Increases Cardiac Contractility in Rats. J Med Chem. 2024 Mar 7.Shipping Conditions:
Room TemperatureClinical Information:
No Development ReportedCAS Number:
2851991-63-2
