PLK1/BRD4-IN-1

CAT: 0931-T64058-01Size: 25 mgDry Ice: NoHazardous: No

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CAT#:0931-T64058-01Size:25 mg

Selected

24/48H Stock Items & 2 to 6 Weeks non Stock Items.

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CAS Number

2412707-81-2

Target

Apoptosis, Androgen Receptor, c-Myc, Epigenetic Reader Domain, PLK, Others

Related Pathways

Cell Cycle/Checkpoint, Others, Endocrinology/Hormones, Apoptosis, Chromatin/Epigenetic

Bioactivity

PLK1/BRD4-IN-1 (9b) is an orally active dual inhibitor of PLK1 (IC50: 22 nM) and BRD4 (IC50: 109 nM) that demonstrates significant anti-tumor efficacy in vivo.

Smiles

C(N1C=2C(N3C([C@H]1CC)=NN=C3C)=CN=C(NC4=C(OC)C=C(C(NC5CCN(C)CC5)=O)C=C4)N2)C6CCCCC6

Molecular Formula

C31H43N9O2

Molecular Weight

573.73

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

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Alternative Products

Catalog	Name
GTR19185523-01	PLK1/BRD4-IN-1
HY-160557-01	PLK1/BRD4-IN-2
HY-160558-01	PLK1/BRD4-IN-3
HY-158031-01	PLK1/BRD4-IN-5
HY-143299	BRD4-BD1-IN-1
HY-161515-01	BRD4/NAMPT-IN-1
MBS5806655	BRD4/CK2-IN-1
GTR19185181-01	PARP1/BRD4-IN-1
MBS5806752	BRD4 D1-IN-1
HY-170841	HDAC3/BRD4-IN-1

PLK1/BRD4-IN-1

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