HDAC3/BRD4-IN-1

CAT: 0931-T205214-01Size: 10 mgDry Ice: NoHazardous: No

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CAT#:0931-T205214-01Size:10 mg

Selected

24/48H Stock Items & 2 to 6 Weeks non Stock Items.

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Target

Epigenetic Reader Domain, HDAC

Related Pathways

DNA Damage/DNA Repair, Chromatin/Epigenetic

Bioactivity

HDAC3/BRD4-IN-1 (compound 26n) is an inhibitor of HDAC3/BRD4, exhibiting an IC50 of 8 nM for HDAC3, while its IC50 values for HDAC1 and HDAC2 are 220 nM and 120 nM, respectively. It displays anti-tumor and anti-proliferative effects by upregulating Ac-H3 and downregulating c-Myc. The half-life of HDAC3/BRD4-IN-1 in human liver microsomes is 29.36 minutes.

Molecular Formula

C31H35N5O4

Molecular Weight

541.64

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

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Catalog	Name
HY-170841	HDAC3/BRD4-IN-1
sc-130319	HDAC3 (1)
BA4164-1	HDAC3-IN-1
HY-161515-01	BRD4/NAMPT-IN-1
HY-143299	BRD4-BD1-IN-1
MBS5806655	BRD4/CK2-IN-1
GTR19185181-01	PARP1/BRD4-IN-1
MBS5806752	BRD4 D1-IN-1
MBS5806722	PLK1/BRD4-IN-1
HY-186002	BRD4/BCL6-IN-1

HDAC3/BRD4-IN-1

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