BRD4-BD1-IN-1

BRD4-BD1-IN-1

• CAS Number: 2761321-18-8
• UNSPSC Description: BRD4-BD1-IN-1 (Compound 9a) is a BRD4-BD1 inhibitor with an IC50 of 38.20 μM[1].
• Target Antigen: Epigenetic Reader Domain
• Type: Reference compound
• Related Pathways: Epigenetics
• Applications: Cancer-programmed cell death
• Field of Research: Cancer
• Assay Protocol: https://www.medchemexpress.com/brd4-bd1-in-1.html
• Solubility: 10 mM in DMSO
• Smiles: CC(OCC1=NC2=C(N1CC3=CC(Br)=CC=C3)C(NC(N2C)=O)=O)=O
• Molecular Weight: 407.22
• References & Citations: [1]Chang Y, et al. Design, synthesis, biological evaluation, and molecular docking of 1, 7-dibenzyl-substituted theophylline derivatives as novel BRD4-BD1-selective inhibitors. Medicinal Chemistry Research, 2021, 30(8): 1453-1468.
• Shipping Conditions: Room temperature
• Clinical Information: No Development Reported