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PARP1/BRD4-IN-2

CAT: 0931-T62540-01Size: 25 mgDry Ice: NoHazardous: No
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CAT#:0931-T62540-01Size:25 mg
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
Quick Request Actions
Target
Others, Apoptosis, PARP, Epigenetic Reader Domain
Related Pathways
Apoptosis, DNA Damage/DNA Repair, Others, Chromatin/Epigenetic
Bioactivity
PARP1/BRD4-IN-2 is a potent and selective inhibitor of PARP1 (IC50: 197 nM) and BRD4 (IC50: 238 nM), which inhibits DNA damage repair, blocks the G0/G1 cell cycle transition, and induces apoptosis. PARP1/BRD4-IN-2 exhibits antitumor effects in the MDA-MB-468 mouse xenograft tumor model and is used to study triple-negative breast cancer (TNBC) .
Molecular Formula
C25H20N4O4
Molecular Weight
440.45
Shipping Conditions
Ice Packs
Storage Temperature
-20°C

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