BRD4-BD1/2-IN-2

BRD4-BD1/2-IN-2

• CAS Number: 2743464-27-7
• UNSPSC Description: BRD4-BD1/2-IN-2 is a potent BRD4 BD2 inhibitor with IC50s of [1].
• Target Antigen: Epigenetic Reader Domain
• Type: Reference compound
• Related Pathways: Epigenetics
• Applications: Cancer-programmed cell death
• Field of Research: Cancer
• Assay Protocol: https://www.medchemexpress.com/brd4-bd1-2-in-2.html
• Solubility: 10 mM in DMSO
• Smiles: O=C(C1=CC(C(C2=CC3=NN(CC(C)(C)O)C=C3C=C2OC4=C(C)C=CC=C4C)=CN5C)=C(N1)C5=O)NCC
• Molecular Weight: 527.61
• References & Citations: [1]Compound functioning as bromodomain protein inhibitor, and composition. WO2021233371A1.
• Shipping Conditions: Room temperature
• Clinical Information: No Development Reported