PROTAC EED degrader-2

CAT: 0931-T12554-01Size: 100 mgDry Ice: NoHazardous: No

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CAT#:0931-T12554-01Size:100 mg

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24/48H Stock Items & 2 to 6 Weeks non Stock Items.

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Target

Histone Methyltransferase, PROTACs

Related Pathways

Chromatin/Epigenetic, PROTAC

Bioactivity

PROTAC EED degrader-2 is a PROTAC targeting EED (pKD of 9.27) and an inhibitor of polycomb repressive complex 2 (PRC2) with a pIC50 of 8.11.

Smiles

FC1=CC=C2C(CCO2)=C1CNC3=NC=C(C4=NN=CN34)C5=C(N=C(C=C5)CCC(NCCCCC(N[C@H](C(N6[C@@H](C[C@H](C6)O)C(NCC7=CC=C(C=C7)C8=C(N=CS8)C)=O)=O)C(C)(C)C)=O)=O)C

Molecular Formula

C50H58FN11O6S

Molecular Weight

960.13

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

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