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PD 156252

CAT: 0804-HY-P10151Size: 1 EachDry Ice: NoHazardous: No
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CAT#:0804-HY-P10151Size:1 Each
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Description
PD 156252 is a hexapeptide that is a highly potent endothelin (ET) antagonist. PD 156252 has enhanced binding affinity for rabbit ETA and rat ETB receptor subtypes with IC50 values of 1.0 and 40 nM, respectively.
CAS Number
175592-65-1
UNSPSC
12352209
Target
Endothelin Receptor
Type
Peptides
Related Pathways
GPCR/G Protein
Applications
Neuroscience-Neuromodulation
Field of Research
Cardiovascular Disease
Assay Protocol
https://www.medchemexpress.com/pd-156252.html
Solubility
10 mM in DMSO
Smiles
OC([C@H](CC1=CNC2=CC=CC=C12)NC([C@H]([C@@H](C)CC)N(C)C([C@H]([C@@H](C)CC)NC([C@H](CC(O)=O)NC([C@H](CC(C)C)NC([C@@H](C3C4=CC=CC=C4CCC5=CC=CC=C53)NC(C)=O)=O)=O)=O)=O)=O)=O
Molecular Formula
C53H69N7O10
Molecular Weight
964.16
References & Citations
[1]Cody WL, et al. Design of a potent combined pseudopeptide endothelin-A/endothelin-B receptor antagonist, Ac-DBhg16-Leu-Asp-Ile-[NMe]Ile-Trp21 (PD 156252) : examination of its pharmacokinetic and spectral properties. J Med Chem. 1997 Jul 4;40 (14) :2228-40.
Shipping Conditions
Room temperature
Scientific Category
Peptides
Clinical Information
No Development Reported

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