Products for Research Use Only
RegisterLogin

RP 72540

CAT: 0804-HY-100481Size: 1 EachDry Ice: NoHazardous: No
Product image 1
1 / 1
CAT#:0804-HY-100481Size:1 Each
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
Quick Request Actions
Description
RP 72540 is a selective CCK-B receptor antagonist, with IC50 values of 2.4, 1.2, and 3.8 nM for CCK-B receptors in the guinea pig cerebral cortex, rat cerebral cortex, and mouse brain, respectively. RP 72540 effectively inhibits CCK-8-induced neuronal firing and dose-dependently inhibits gastric acid secretion, making it potentially valuable in studies of acid secretion. RP 72540 is an important tool for investigating the physiological functions of CCK B receptors[1].
CAS Number
139088-45-2
Product Name Alternative
RPR101048
UNSPSC
12352005
Target
Cholecystokinin Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/rp-72540.html
Smiles
O=C(N(C1=CC=CC(OC)=C1)CC(N(C)C2=CC=CC=C2)=O)CNC(NC3=CC=CC(C(C(O)=O)C)=C3)=O
Molecular Formula
C28H30N4O6
Molecular Weight
518.56
References & Citations
[1]Bertrand P, et al. Pharmacological properties of ureido-acetamides, new potent and selective non-peptide CCKB/gastrin receptor antagonists. Eur J Pharmacol. 1994 Sep 12;262 (3) :233-45.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported

Related Products

CatalogName
HY-101939RP-001
HY-P11107-01RP-832c
HY-172737-01RP-1664
HY-116260RP-69758
HY-108483-01RP 67580
HY-100530ARp-cAMPS
HY-10015348740 RP
HY-100160RP 54275
HY-P5565RP-1
HY-158346RP-2119

Alternative Products

CatalogName
T28612-01RP-72540

Popular Products