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RP-72540

CAT: 0931-T28612-01Size: 25 mgDry Ice: NoHazardous: No
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CAT#:0931-T28612-01Size:25 mg
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
139088-45-2
Target
Cholecystokinin Receptor, Others
Related Pathways
Others, GPCR/G Protein
Bioactivity
RP-72540 is a cholecystokinin B receptor antagonist. RP 72540 showed selectivity factors in express of 200 for CCKA versus CCKB receptors and also had high affinity for gastrin binding sites in the stomach. Administration of RP-72540 resulted in a dose-dependent inhibition of [3H]pCCK-8 binding in mouse brain homogenate. However, the relative penetration of RP-72540 into the forebrain after peripheral administration was below 0.01%.
Smiles
N(CC(N(C)C1=CC=CC=C1)=O)(C(CNC(NC2=CC(C(C(O)=O)C)=CC=C2)=O)=O)C3=CC(OC)=CC=C3
Molecular Formula
C28H30N4O6
Molecular Weight
518.56
Shipping Conditions
Ice Packs
Storage Temperature
-20°C

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