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PKR activator 5

CAT: 0804-HY-159095Size: 1 EachDry Ice: NoHazardous: No
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CAT#:0804-HY-159095Size:1 Each
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
PKR activator 5 (Compound 18) is an activator for pyruvate kinase R (PKR) with an AC50 of 28 nM[1].
CAS Number
2761226-35-9
UNSPSC
12352005
Target
Pyruvate Kinase
Type
Reference compound
Related Pathways
Metabolic Enzyme/Protease
Field of Research
Others
Assay Protocol
https://www.medchemexpress.com/pkr-activator-5.html
Smiles
CC1=NN(C(CNC(NCC2=NC=NN2C3=CC4=C(C=C3)C=CC=N4)=O)=N1)C5=CC=C(C(F)=C5)Cl
Molecular Formula
C23H19ClFN9O
Molecular Weight
491.91
References & Citations
[1]Yu C, et al., The search for pyruvate kinase-R activators; from a HTS screening hit via an impurity to the discovery of a lead series. Bioorg Med Chem Lett. 2024 Jun 29;110:129865.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported

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