CHIR-2279

• UNSPSC Description:

  CHIR-2279 is a high-affinity ligand (Ki=5 nM) for the α1-adrenergic receptor and can be further studied as a drug lead compound[1].

• Target Antigen:

  Adrenergic Receptor

• Type:

  Reference compound

• Related Pathways:

  GPCR/G Protein;Neuronal Signaling

• Field of Research:

  Others

• Assay Protocol:

  https://www.medchemexpress.com/chir-2279.html

• Smiles:

  O=C(CN(CCC1=CC=CC=C1)C(CN(C(CNCCC2=CC=C(C=C2)O)=O)C3=CC=C(C4=CC=CC=C4)C=C3)=O)N

• Molecular Weight:

  564.67

• References & Citations:

  [1]Zuckermann, et al. Discovery of nanomolar ligands for 7-transmembrane G-protein-coupled receptors from a diverse N-(substituted) glycine peptoid library. Journal of medicinal chemistry 37.17 (1994): 2678-2685.

• Shipping Conditions:

  Room temperature

• Clinical Information:

  No Development Reported

• CAS Number:

  158198-45-9