Products for Research Use Only

CHIR 4531

CAT: 0804-HY-120846Size: 1 EachDry Ice: NoHazardous: No
Product image 1
1 / 1
CAT#:0804-HY-120846Size:1 Each
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
Quick Request Actions
Description
CHIR 4531, a trimer peptide, is a opiate ligand that binds to the mu-opiate receptor with a Ki of 6 nM[1].
CAS Number
158198-48-2
UNSPSC
12352005
Target
Opioid Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/chir-4531.html
Smiles
O=C(N)CN(C(CN(C(CNCC(C1=CC=CC=C1)C2=CC=CC=C2)=O)CC3=CC=C(OCO4)C4=C3)=O)CCC5=CC=C(O)C=C5
Molecular Formula
C36H38N4O6
Molecular Weight
622.71
References & Citations
[1]R N Zuckermann, et al. Discovery of nanomolar ligands for 7-transmembrane G-protein-coupled receptors from a diverse N- (substituted) glycine peptoid library. J Med Chem. 1994 Aug 19;37 (17) :2678-85.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
μ Opioid Receptor/MOR