THR-β agonist 7

CAT: 0804-HY-160266Size: 1 mgDry Ice: NoHazardous: No

CAT#:0804-HY-160266Size:1 mg

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Description

THR-β agonist-1 (Example 2) is a THR-β agonist, with EC50 values of 52 nM and 1017 nM for THR-β and THR-α, respectively[1].

CAS Number

[2604229-32-3]

UNSPSC

12352005

Target

Thyroid Hormone Receptor

Type

Isotope-Labeled Compounds

Related Pathways

Vitamin D Related/Nuclear Receptor

Applications

Metabolism-protein/nucleotide metabolism

Field of Research

Cancer; Metabolic Disease

Solubility

10 mM in DMSO

Smiles

O=C1N(C2=CC(Br)=C(C(Cl)=C2)OC(C=C3C(C([2H])([2H])[2H])C([2H])([2H])[2H])=NNC3=O)N=C(C(N1)=O)C#N

Molecular Formula

C17H6D6BrClN6O4

Molecular Weight

485.71

References & Citations

[1], et al. Halogen-substituted phenylate compound and applications thereof. Patent WO2021032161A1.

Shipping Conditions

Room temperature

Scientific Category

Isotope-Labeled Compounds

Clinical Information

No Development Reported

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