DPP-4-IN-9

• UNSPSC Description:

  DPP-4-IN-9 (compound 6l) is a potent inhibitor of dipeptidyl peptidase DPP-4 (IC50: 8.22 nM). DPP-4-IN-9 has antihyperglycemic activity[1].

• Target Antigen:

  Dipeptidyl Peptidase

• Type:

  Reference compound

• Related Pathways:

  Metabolic Enzyme/Protease

• Applications:

  Metabolism-protein/nucleotide metabolism

• Field of Research:

  Metabolic Disease

• Assay Protocol:

  https://www.medchemexpress.com/dpp-4-in-9.html

• Solubility:

  10 mM in DMSO

• Smiles:

  O=C(N/N=C/C1=CC=C(OC)C(OC)=C1)CN2C(C(C#N)=C(C3=CC=CC=C3)C(C4=CC=CC=C4)=N2)=O

• Molecular Weight:

  493.51

• References & Citations:

  [1]Nidhar M, et al. Ligand-based designing of DPP-4 inhibitors via hybridization; synthesis, docking, and biological evaluation of pyridazine-acetohydrazides. Mol Divers. 2023 Dec;27(6):2729-2740.

• Shipping Conditions:

  Room temperature

• Clinical Information:

  No Development Reported

• CAS Number:

  2906243-39-6