DPP-4-IN-9

• Description:

  DPP-4-IN-9 (compound 6l) is a potent inhibitor of dipeptidyl peptidase DPP-4 (IC50: 8.22 nM) . DPP-4-IN-9 has antihyperglycemic activity[1].

• UNSPSC:

  12352005

• Target:

  Dipeptidyl Peptidase

• Type:

  Reference compound

• Related Pathways:

  Metabolic Enzyme/Protease

• Applications:

  Metabolism-protein/nucleotide metabolism

• Field of Research:

  Metabolic Disease

• Assay Protocol:

  https://www.medchemexpress.com/dpp-4-in-9.html

• Solubility:

  10 mM in DMSO

• Smiles:

  O=C (N/N=C/C1=CC=C (OC) C (OC) =C1) CN2C (C (C#N) =C (C3=CC=CC=C3) C (C4=CC=CC=C4) =N2) =O

• Molecular Formula:

  C28H23N5O4

• Molecular Weight:

  493.51

• References & Citations:

  [1]Nidhar M, et al. Ligand-based designing of DPP-4 inhibitors via hybridization; synthesis, docking, and biological evaluation of pyridazine-acetohydrazides. Mol Divers. 2023 Dec;27 (6) :2729-2740.

• Shipping Conditions:

  Room temperature

• Scientific Category:

  Reference compound1

• Clinical Information:

  No Development Reported

• CAS Number:

  2906243-39-6