BuChE-IN-4

CAT: 0804-HY-146687Size: 1 EachDry Ice: NoHazardous: No
CAT#:0804-HY-146687Size:1 Each
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Description
BuChE-IN-4 (Compound C6) is a potent inhibitor of BuChE with an IC50 of 7.7 nM. BuChE-IN-4 exhibits mild antioxidant capacity, nontoxicity, lipophilicity and neuroprotective activity[1].
CAS Number
[2499490-52-5]
UNSPSC
12352005
Target
Cholinesterase (ChE)
Type
Reference compound
Related Pathways
Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/buche-in-4.html
Solubility
10 mM in DMSO
Smiles
O=S1(CCC2=C(N(N=C2CN(CC3=CC=C(C=C3)Br)CCO)C4=CC=CC=C4F)O1)=O
Molecular Formula
C21H21BrFN3O4S
Molecular Weight
510.38
References & Citations
[1]Zhang Z, et al. The structure-based optimization of δ-sultone-fused pyrazoles as selective BuChE inhibitors. Eur J Med Chem. 2020 Sep 1;201:112273.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
BChE

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