BRD4-BD1/2-IN-1

BRD4-BD1/2-IN-1

• CAS Number: 1781219-19-9
• UNSPSC Description: BRD4-BD1/2-IN-1 is a potent BRD4 inhibitor with IC50s of [1].
• Target Antigen: Epigenetic Reader Domain
• Type: Reference compound
• Related Pathways: Epigenetics
• Applications: Cancer-programmed cell death
• Field of Research: Cancer
• Assay Protocol: https://www.medchemexpress.com/brd4-bd1-2-in-1.html
• Solubility: 10 mM in DMSO
• Smiles: O=C1C2=C(C(C3=CC4=C(C=C3OC5=CC=C(C=C5F)F)N=CN4)=CN1C)C=CN2
• Molecular Weight: 392.36
• References & Citations: [1]Bicyclic heterocycles as bet protein inhibitors. US20150148375A1.
• Shipping Conditions: Room temperature
• Clinical Information: No Development Reported