EZH2-IN-5

EZH2-IN-5

• CAS Number: 1403258-69-4
• UNSPSC Description: EZH2-IN-5 is a potent EZH2 inhibitor with IC50 values of 1.52 nM and 4.07 nM for wild-type and mutant Tyr641 EZH2, respectively[1].
• Target Antigen: Histone Methyltransferase
• Type: Reference compound
• Related Pathways: Epigenetics
• Applications: Cancer-programmed cell death
• Field of Research: Cancer
• Assay Protocol: https://www.medchemexpress.com/ezh2-in-5.html
• Solubility: 10 mM in DMSO
• Smiles: CCN([C@H]1CC[C@@H](CC1)N(C)C)C2=C(C(C(NCC3=C(C=C(NC3=O)C)C)=O)=CC(Br)=C2)C
• Molecular Weight: 517.50
• References & Citations: [1]Richard Chesworth, et al. Substituted benzene compounds. WO2012142513A1
• Shipping Conditions: Room temperature
• Clinical Information: No Development Reported