EZH2-IN-5
CAT:
804-HY-141566
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- Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
- Dry Ice Shipment: No
EZH2-IN-5
- CAS Number: 1403258-69-4
- UNSPSC Description: EZH2-IN-5 is a potent EZH2 inhibitor with IC50 values of 1.52 nM and 4.07 nM for wild-type and mutant Tyr641 EZH2, respectively[1].
- Target Antigen: Histone Methyltransferase
- Type: Reference compound
- Related Pathways: Epigenetics
- Applications: Cancer-programmed cell death
- Field of Research: Cancer
- Assay Protocol: https://www.medchemexpress.com/ezh2-in-5.html
- Solubility: 10 mM in DMSO
- Smiles: CCN([C@H]1CC[C@@H](CC1)N(C)C)C2=C(C(C(NCC3=C(C=C(NC3=O)C)C)=O)=CC(Br)=C2)C
- Molecular Weight: 517.50
- References & Citations: [1]Richard Chesworth, et al. Substituted benzene compounds. WO2012142513A1
- Shipping Conditions: Room temperature
- Clinical Information: No Development Reported