EZH2-IN-2

CAT: 0804-HY-A0298-01Size: 5 mgDry Ice: NoHazardous: No
CAT#:0804-HY-A0298-01Size:5 mg
Selected
PRICE
AVAILABILITY: InStock
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
Product image 1
1 / 1
Description
EZH2-IN-2 (Example 69) is a EZH2 inhibitor with an IC50 and a TR-FRET IC50 of 64 nM and 20 nM. EZH2-IN-2 can be used for the research of cancer or precancerous condition related to EZH2 activity[1].
CAS Number
[2238821-31-1]
UNSPSC
12352005
Target
Histone Methyltransferase
Type
Reference compound
Related Pathways
Epigenetics
Applications
Cancer-programmed cell death
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/ezh2-in-2.html
Purity
99.60
Solubility
DMSO : 10 mg/mL (ultrasonic; warming; heat to 60°C)
Smiles
O=C(NCC1=C(C)C=C(C)NC1=O)C2=CC(C3=CC=C(N4CCN(CC5CC5)CC4)N=C3C)=CC(N(C(C6CC6)=O)CC)=C2C
Molecular Formula
C36H46N6O3
Molecular Weight
610.79
References & Citations
[1]LIU, Qing Song, et al. Ezh2 inhibitor and use thereof. WO2018133795A1.
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
EZH2

Related Products

CatalogName
HY-149463EZH2-IN-16
HY-P2266-01SAH-EZH2
HY-144096EZH2-IN-11
HY-149726-01EZH2-IN-17
HY-148458-01EZH2-IN-14
HY-141566EZH2-IN-5
HY-174372EZH2-IN-23
HY-D2274EZH2-AF647
HY-161419EZH2-IN-18
HY-169958EZH2-IN-22

Alternative Products

CatalogName
BA4850-5.1EZH2-IN-2
462249EZH2-​IN-​2
MF-0116331-01PARP/EZH2-IN-2
E9085-02LEZH2 (Protein Ezh2) discontinued
E8EM1706-15EZH2
A23982-1PROTAC EZH2 Degrader-2 1mg
A23982-5PROTAC EZH2 Degrader-2 5mg
A23982-10PROTAC EZH2 Degrader-2 10mg
A23982-50PROTAC EZH2 Degrader-2 50mg
BNUM2536-50EZH2 / KMT6 (EZH2/2536), 1mg/mL

Popular Products