PDE1-IN-3
CAT:
804-HY-130262
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- Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
- Dry Ice Shipment: No


PDE1-IN-3
UNSPSC Description:
PDE1-IN-3, compound 4 (WO2019156861), is a selective human phosphodiesterase 1 (PDE1) inhibitor. PDE1-IN-3 inhibits PDE4D and PDE6AB with IC50 values of 23.99 μM and 10 μM, respectively[1].Target Antigen:
Phosphodiesterase (PDE)Type:
Reference compoundRelated Pathways:
Metabolic Enzyme/ProteaseApplications:
COVID-19-immunoregulationField of Research:
Inflammation/ImmunologyAssay Protocol:
https://www.medchemexpress.com/pde1-in-3.htmlSolubility:
10 mM in DMSOSmiles:
O=C1C2=NN=C(C3(C4CC4)CC3)N2C(C)=C(C)N1CC5CCC5Molecular Weight:
312.41References & Citations:
[1]Nicholas Paul Camp, et al. [1,2,4]triazolo[4,3-a]pyrazin-8-one derivativesShipping Conditions:
Room temperatureClinical Information:
No Development ReportedCAS Number:
2370966-46-2