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ENMD-1068 (hydrobromide)

CAT: 0804-HY-122049Size: 1 EachDry Ice: NoHazardous: No
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CAT#:0804-HY-122049Size:1 Each
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Description
ENMD-1068 hydrobromide is a potent PAR2 antagonist. ENMD-1068 hydrobromide attenuates joint inflammation in a dose-dependent manner. ENMD-1068 hydrobromide can be used in research of joint inflammation[1].
CAS Number
644961-61-5
UNSPSC
12352005
Target
Protease Activated Receptor (PAR)
Type
Reference compound
Related Pathways
GPCR/G Protein
Applications
COVID-19-immunoregulation
Field of Research
Inflammation/Immunology
Assay Protocol
https://www.medchemexpress.com/enmd-1068-hydrobromide.html
Solubility
10 mM in DMSO
Smiles
O=C(N1CCN(C(CC(C)C)=O)CC1)CCCCCN.Br
Molecular Formula
C15H30BrN3O2
Molecular Weight
364.32
References & Citations
[1]Kelso EB, et, al. Therapeutic promise of proteinase-activated receptor-2 antagonism in joint inflammation. J Pharmacol Exp Ther. 2006 Mar;316 (3) :1017-24.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
PAR2