ENMD-1068 (hydrobromide)

ENMD-1068 (hydrobromide)

• CAS Number: 644961-61-5
• UNSPSC Description: ENMD-1068 hydrobromide is a potent PAR2 antagonist. ENMD-1068 hydrobromide attenuates joint inflammation in a dose-dependent manner. ENMD-1068 hydrobromide can be used in research of joint inflammation[1].
• Target Antigen: Protease Activated Receptor (PAR)
• Type: Reference compound
• Related Pathways: GPCR/G Protein
• Applications: COVID-19-immunoregulation
• Field of Research: Inflammation/Immunology
• Assay Protocol: https://www.medchemexpress.com/enmd-1068-hydrobromide.html
• Solubility: 10 mM in DMSO
• Smiles: O=C(N1CCN(C(CC(C)C)=O)CC1)CCCCCN.Br
• Molecular Weight: 364.32
• References & Citations: [1]Kelso EB, et, al. Therapeutic promise of proteinase-activated receptor-2 antagonism in joint inflammation. J Pharmacol Exp Ther. 2006 Mar;316(3):1017-24.
• Shipping Conditions: Room temperature
• Clinical Information: No Development Reported