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BMS-986163

CAT: 0804-HY-107774Size: 1 EachDry Ice: NoHazardous: No
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CAT#:0804-HY-107774Size:1 Each
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Description
BMS-986163 is a negative allosteric modulator of GluN2B. The proagent BMS-986163 rapidly converts to its active parent molecule BMS-986169 (Ki=4 nM, IC50=24 nM) .
CAS Number
1801151-09-6
UNSPSC
12352005
Target
IGluR
Type
Reference compound
Related Pathways
Membrane Transporter/Ion Channel; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/BMS-986163.html
Solubility
10 mM in DMSO
Smiles
CC1=CC=C(CN2CC[C@@H](N3C[C@@H](F)[C@H](C4=CC=C(OP(O)(O)=O)C=C4)CC3)C2=O)C=C1
Molecular Formula
C23H28FN2O5P
Molecular Weight
462.45
References & Citations
[1]Marcin LR, et al. BMS-986163, a Negative Allosteric Modulator of GluN2B with Potential Utility in Major Depressive Disorder. ACS Med Chem Lett. 2018 Apr 13;9 (5) :472-477.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported

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