TUG-2099

• UNSPSC Description:

  TUG-2099 (compound 4s) is a potent GPR84 agonist with the EC50 of 0.3 nM. TUG-2099 can be used for study of Alzheimer’s disease, atherosclerosis, cancer, and so an[1].

• Target Antigen:

  GPR84

• Type:

  Reference compound

• Related Pathways:

  GPCR/G Protein

• Applications:

  Cancer-programmed cell death

• Field of Research:

  Cancer; Neurological Disease; Cardiovascular Disease

• Assay Protocol:

  https://www.medchemexpress.com/tug-2099.html

• Solubility:

  10 mM in DMSO

• Smiles:

  CCCC1=CC=C(C=C1)CCC2=CC(O)=CC(N2)=O

• Molecular Weight:

  257.33

• References & Citations:

  [1]Ieremias L, et al. Structure-Activity Relationship Studies and Optimization of 4-Hydroxypyridones as GPR84 Agonists. J Med Chem. Published online February 21, 2024.

• Shipping Conditions:

  Room temperature

• Clinical Information:

  No Development Reported