PKM2-IN-9

• Description:

  PKM2-IN-9 (compound C1) is a potent inhibitor of PKM2, with the inhibition rate of 75% at 50 μM. PKM2-IN-9 plays an important role in cancer research[1].

• UNSPSC:

  12352005

• Target:

  Pyruvate Kinase

• Related Pathways:

  Metabolic Enzyme/Protease

• Field of Research:

  Cancer

• Smiles:

  O=C(C1=CC=CC=C1)NCC2=NC3=C(N2CC(NC4=CC=CC(C)=C4)=O)C=CC=C3

• Molecular Formula:

  C24H22N4O2

• Molecular Weight:

  398.46

• References & Citations:

  [1]Beth Israel Deaconess Medical Center. Pyruvate kinase M2 inhibitors and methods using them for the treatment of disease. World Intellectual Property Organization, WO2008019139 A2 2008-02-14

• Shipping Conditions:

  Room temperature

• Scientific Category:

  Reference compound1

• Clinical Information:

  No Development Reported

• CAS Number:

  [498568-75-5]