SAS-1121

• Description:

  SAS-1121 is a subtype-selective sigma 2 receptor/PGRMC1 ligand with a Ki of 16.2 nM. SAS-1121 is 574-fold selective for the signma 2 receptor over the sigma 1 receptor. SAS-1121 is a tertiary amine. SAS-1121 can be studied in neurology-related research[1].

• UNSPSC:

  12352005

• Target:

  Sigma Receptor

• Related Pathways:

  Neuronal Signaling

• Applications:

  Neuroscience-Neuromodulation

• Field of Research:

  Neurological Disease

• Smiles:

  O=C(N1CC[C@]2([H])C3=CC=C(N4CCN(CCC(OCC)=O)CC4)C=C3[C@@]1([H])C2)OCC5=CC=CC=C5

• Molecular Formula:

  C28H35N3O4

• Molecular Weight:

  477.60

• References & Citations:

  [1]Sahn, J. J., et al., (2016) . Norbenzomorphan Framework as a Novel Scaffold for Generating Sigma 2 Receptor/PGRMC1 Subtype-Selective Ligands. ChemMedChem, 11 (6), 556-561.

• Shipping Conditions:

  Room temperature

• Scientific Category:

  Reference compound1

• Clinical Information:

  No Development Reported

• CAS Number:

  [2095551-67-8]