Cibenzoline succinate

• Target:

  Potassium Channel

• Related Pathways:

  Membrane transporter/Ion channel

• Bioactivity:

  Cibenzolinesuccinate (Cifenline succinate) is the succinate salt form of Cibenzoline. It serves as an inhibitor of ATP-sensitive potassium channels (KATP), affecting the Kir6.2 subunit, with an IC50 of 22.2 µM. This compound influences insulin secretion and exhibits both antiarrhythmic and antidiabetic properties.

• Smiles:

  O=C(O)CCC(=O)O.N1=C(NCC1)C2CC2(C=3C=CC=CC3)C=4C=CC=CC4

• Molecular Formula:

  C22H24N2O4

• Molecular Weight:

  380.44

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C

• CAS Number:

  100678-32-8